Synthesis of Thieno [2, 3-d] pyrimidine Derivatives and Their Antifungal Activities
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چکیده
منابع مشابه
Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
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An electroorganic reaction for the synthesis of 7-amino-2, 4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-pyrano[2, 3-d] pyrimidine-6-carbonitrile and ethyl-7-amino-2, 4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-pyrano[2, 3-d] pyrimidine-6-carboxylate derivatives are described, using an electrogenerated base of the anion of malonitrile or ethylcyanoacetate. This one-pot, three-component condensation of an a...
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ژورنال
عنوان ژورنال: YAKUGAKU ZASSHI
سال: 1989
ISSN: 0031-6903,1347-5231
DOI: 10.1248/yakushi1947.109.7_464